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Back Cover: Potent and Selective Inhibitors of Trypanosoma cruzi Triosephosphate Isomerase with Concomitant Inhibition of Cruzipain: Inhibition of Parasite Growth through Multitarget Activity (ChemMedChem 12/2016)
Aguilera, Elena ; Varela, Javier ; Birriel, Estefanía ; Serna, Elva ; Torres, Susana ; Yaluff, Gloria ; de Bilbao, Ninfa Vera ; Aguirre‐López, Beatriz ; Cabrera, Nallely ; Díaz Mazariegos, Selma ; de Gómez‐Puyou, Marieta Tuena ; Gómez‐Puyou, Armando ; Pérez‐Montfort, Ruy ; Minini, Lucia ; Merlino, Alicia ; Cerecetto, Hugo ; González, Mercedes ; Alvarez, Guzmán
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Multifunctional, Fluorene‐Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease
Panek, Dawid ; Pasieka, Anna ; Jończyk, Jakub ; Gawlińska, Milena ; Zaręba, Paula ; Siwek, Agata ; Wolak, Małgorzata ; Mordyl, Barbara ; Głuch‐Lutwin, Monika ; Latacz, Gniewomir ; Brazzolotto, Xavier ; Chantegreil, Fabien ; Nachon, Florian ; Zdarova Karasova, Jana ; Pejchal, Jaroslav ; Mzik, Martin ; Sestak, Vit ; Prchal, Lukas ; Odvarkova, Jitka ; Soukup, Ondrej ; Korabecny, Jan ; Sorf, Ales ; Hamsikova, Marie ; Zemanova, Lucie ; Muckova, Lubica ; Vánova, Nela ; Dryja, Pola ; Sałat, Kinga ; Höfner, Ge
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Multifunctional, Fluorene‐Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease
Panek, Dawid ; Pasieka, Anna ; Jończyk, Jakub ; Gawlińska, Milena ; Zaręba, Paula ; Siwek, Agata ; Wolak, Małgorzata ; Mordyl, Barbara ; Głuch‐Lutwin, Monika ; Latacz, Gniewomir ; Brazzolotto, Xavier ; Chantegreil, Fabien ; Nachon, Florian ; Zdarova Karasova, Jana ; Pejchal, Jaroslav ; Mzik, Martin ; Sestak, Vit ; Prchal, Lukas ; Odvarkova, Jitka ; Soukup, Ondrej ; Korabecny, Jan ; Sorf, Ales ; Hamsikova, Marie ; Zemanova, Lucie ; Muckova, Lubica ; Vánova, Nela ; Dryja, Pola ; Sałat, Kinga ; Höfner, Ge
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Synthesis, Antiplasmodial, and Antileukemia Activity of Dihydroartemisinin–HDAC Inhibitor Hybrids as Multitarget Drugs
von Bredow, Lukas ; Schäfer, Thomas Martin ; Hogenkamp, Julian ; Tretbar, Maik ; Stopper, Daniel ; Kraft, Fabian B. ; Schliehe-Diecks, Julian ; Schöler, Andrea ; Borkhardt, Arndt ; Bhatia, Sanil ; Held, Jana ; Hansen, Finn Kristian 2023 Universitätsbibliothek Leipzig
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Multitarget Drugs: Synthesis and Preliminary Pharmacological Characterization of Zileuton Analogues Endowed with Dual 5‐LO Inhibitor and NO‐Dependent Activities
Boschi, Donatella ; Giorgis, Marta ; Cena, Clara ; Talniya, Naveen Chandra ; Di Stilo, Antonella ; Morini, Giuseppina ; Coruzzi, Gabriella ; Guaita, Elena ; Fruttero, Roberta ; Gasco, Alberto
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Multitarget‐Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H 3 R Antagonism for Neurodegenerative Diseases
Bautista‐Aguilera, Óscar M. ; Hagenow, Stefanie ; Palomino‐Antolin, Alejandra ; Farré‐Alins, Víctor ; Ismaili, Lhassane ; Joffrin, Pierre‐Louis ; Jimeno, María L. ; Soukup, Ondřej ; Janočková, Jana ; Kalinowsky, Lena ; Proschak, Ewgenij ; Iriepa, Isabel ; Moraleda, Ignacio ; Schwed, Johannes S. ; Romero Martínez, Alejandro ; López‐Muñoz, Francisco ; Chioua, Mourad ; Egea, Javier ; Ramsay, Rona R. ; Marco‐Contelles, José ; Stark, Holger
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11‐Substituted Benzo (c) phenanthridines: New Structures and Insight into Their Mode of Antiproliferative Action
Clement, Bernd ; Girreser, Ulrich ; Steinhauer, Tamara N. ; Meier, Christopher ; Marko, Doris ; Aichinger, Georg ; Kaltefleiter, Ilka ; Stenzel, Lars ; Heber, Dieter ; Weide, Matthias ; Wolschendorf, Ulrich ; Zebothsen, Inga ; zur Nieden, Dana
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Systematic Assessment of Fragment Identification for Multitarget Drug Design
Brunst, Steffen ; Kramer, Jan S. ; Kilu, Whitney ; Heering, Jan ; Pollinger, Julius ; Hiesinger, Kerstin ; George, Sven ; Steinhilber, Dieter ; Merk, Daniel ; Proschak, Ewgenij
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Corrigendum: Designing Multitarget Anti‐inflammatory Agents: Chemical Modulation of the Lumiracoxib Structure toward Dual Thromboxane Antagonists–COX‐2 Inhibitors
Bertinaria, Massimo ; Shaikh, Mohammed Abrar Abdul Gaffar ; Buccellati, Carola ; Cena, Clara ; Rolando, Barbara ; Lazzarato, Loretta ; Fruttero, Roberta ; Gasco, Alberto ; Hoxha, Malvina ; Capra, Valérie ; Sala, Angelo ; Rovati, G. Enrico
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Focused design of polypharmacophoric neuroprotective compounds: Conjugates of γ-carbolines with carbazole derivatives and tetrahydrocarbazole
Makhaeva, Galina F. ; Sokolov, Vladimir B. ; Shevtsova, Elena F. ; Kovaleva, Nadezhda V. ; Lushchekina, Sofya V. ; Boltneva, Natalia P. ; Rudakova, Elena V. ; Aksinenko, Alexey Yu. ; Shevtsov, Pavel N. ; Neganova, Margarita E. ; Dubova, Ludmila G. ; Bachurin, Sergey O.
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Multitarget drugs: Focus on the NO-donor hybrid drugs
Gasco, Alberto ; Boschi, Donatella ; Chegaev, Konstantin ; Cena, Clara ; Di Stilo, Antonella ; Fruttero, Roberta ; Lazzarato, Loretta ; Rolando, Barbara ; Tosco, Paolo
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A Multitargeted Approach to Breast Cancer Therapy: Exploring the Therapeutic Potential of Afzelin as a Combination Agent with FDA-Approved Breast Cancer Drugs
Francis, Dhilna ; T G, Abi ; R N, Binitha
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Recent Insights in Multi‐Target Drugs in Pharmacology and Medicinal Chemistry
Cemali, Sadık Hüseyin ; Poyraz, Samet ; Belveren, Samet ; Taş, Senanur ; Tamer, Mehmet Ali ; Döndaş, Naciye Yaktubay ; Döndaş, H. Ali ; Sansano, Jose Miguel
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Contilistat, a New Multitarget Small Polyfunctionalized Indole Derivative
Toledano-Pinedo, Mireia ; Diez-Iriepa, Daniel ; Porro-Pérez, Alicia ; Schäker-Hübner, Linda ; Hanl, Maria ; Samadi, Abdelouahid ; Almendros, Pedro ; Iriepa, Isabel ; Rodríguez-Fernández, M. Mercedes ; Griñán-Ferré, Christian ; Siwek, Agata ; Wolak, Małgorzata ; Satała, Grzegorz ; Bojarski, Andrzej J. ; Doroż-Płonka, Agata ; Handzlik, Jadwiga ; Godyń, Justyna ; Knez, Damijan ; Gobec, Stanislav ; Więckowska, Anna ; Hansen, Finn Kristian ; Marco-Contelles, José
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Identification of 2,4‐Dinitro‐Biphenyl‐Based Compounds as MAPEG Inhibitors
Di Micco, Simone ; Terracciano, Stefania ; Pierri, Martina ; Cantone, Vincenza ; Liening, Stefanie ; König, Stefanie ; Garscha, Ulrike ; Hofstetter, Robert Klaus ; Koeberle, Andreas ; Werz, Oliver ; Bruno, Ines ; Bifulco, Giuseppe
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8‐Benzyltetrahydropyrazino (2,1‐ f) purinediones: Water‐Soluble Tricyclic Xanthine Derivatives as Multitarget Drugs for Neurodegenerative Diseases
Brunschweiger, Andreas ; Koch, Pierre ; Schlenk, Miriam ; Pineda, Felipe ; Küppers, Petra ; Hinz, Sonja ; Köse, Meryem ; Ullrich, Stefan ; Hockemeyer, Jörg ; Wiese, Michael ; Heer, Jag ; Müller, Christa E.
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In vitro cytostatic effect on tumor cells by carborane-based dual cyclooxygenase-2 and 5-lipoxygenase inhibitors
Braun, Sebastian ; Paskas, Svetlana ; Laube, Markus ; George, Sven ; Hofmann, Bettina ; Lönnecke, Peter ; Steinhilber, Dieter ; Pietzsch, Jens ; Mijatović, Sanja S. ; Maksimović-Ivanić, Danijela ; Hey-Hawkins, Evamarie 2022 Universitätsbibliothek Johann Christian Senckenberg
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Selective Estrogen Receptor Modulators – A New Brand of Multitarget Drugs
Cano, Antonio 2006 Springer Berlin
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Systematic assessment of fragment identification for multitarget drug design
Brunst, Steffen ; Kramer, Jan S. ; Kilu, Whitney ; Heering, Jan ; Pollinger, Julius ; Hiesinger, Kerstin ; George, Sven ; Steinhilber, Dieter ; Merk, Daniel ; Proschak, Ewgenij 2020 Universitätsbibliothek Johann Christian Senckenberg
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Multitarget drugs in cancer therapy - carborane-based dual COX-2/5-LO inhibitors
Braun, Sebastian 2023